SCHEMBL16309355

SCHEMBL16309355

Cc1ccc(C2(C(=O)Nc3ccc4[nH]c(C(C)(C)C)cc4c3)CC2)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CFTR P13569 6/20 0.54
MAOA P21397 4/20 0.41
MAOB P27338 4/20 0.41
THRB P10828 1/20 0.40
PTGES O14684 2/20 0.39
HPGD P15428 2/20 0.39
HDAC1 Q13547 1/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NR2E3 Q9Y5X4 1/20 0.38
ACKR3 P25106 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14403601 0.92 CFTR (0.54) CFTRMAOAMAOBHDAC1NR2E3
SCHEMBL12741876 0.92 CFTR (0.56) CFTRMAOAMAOBHDAC1POLB
SCHEMBL12741871 0.90 CFTR (0.54) CFTRMAOAMAOBHDAC1NR2E3
SCHEMBL12741525 0.89 CFTR (0.55) CFTRMAOAMAOBHDAC1NR2E3
SCHEMBL12741439 0.89 CFTR (0.58) CFTRMAOAMAOBHDAC1ALDH1A1
SCHEMBL20194957 0.88 CFTR (0.54) CFTRMAOAMAOBHDAC1ALDH1A1
SCHEMBL20195007 0.88 CFTR (0.54) CFTRMAOAMAOBHDAC1
SCHEMBL12741332 0.87 CFTR (0.58) CFTRMAOBHPGDHDAC1POLB
SCHEMBL19753053 0.87 CFTR (0.55) CFTRMAOAMAOBHPGDHDAC1
SCHEMBL12741185 0.87 CFTR (0.56) CFTRMAOAMAOBTHRBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8912199-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-12-16 US disclosed