SCHEMBL16319574

SCHEMBL16319574

Cc1cc(C)c(CNC(=O)c2cc(C3CC3)nc3c2cnn3CCN(C(=O)O)C(C)(C)C)c(=O)[nH]1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 20/20 0.66
EED O75530 3/20 0.66
RBBP4 Q09028 3/20 0.66
SUZ12 Q15022 3/20 0.66
RBBP7 Q16576 2/20 0.66
AEBP2 Q6ZN18 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12503369 0.87 EZH2 (0.72) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL10255119 0.87 EZH2 (0.76) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL1695112 0.86 EZH2 (0.73) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL10254671 0.85 EZH2 (0.79) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL10254889 0.84 EZH2 (0.66) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL10254852 0.83 EZH2 (0.69) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL10255280 0.81 EZH2 (0.78) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL12499687 0.80 EZH2 (1.00) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL14755009 0.78 EZH2 (0.86) EZH2EEDRBBP4SUZ12RBBP7
SCHEMBL10256868 0.77 EZH2 (0.73) EZH2EEDRBBP4SUZ12RBBP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566479-B1 AZAINDAZOLES GLAXOSMITHKLINE LLC (US) 2014-12-24 EP disclosed