SCHEMBL16341908

SCHEMBL16341908

Cc1ccc(OC(c2cccc(Cl)c2)c2cc(-c3ccc(CN4CC(C(=O)O)C4)cc3)no2)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.53
S1PR5 Q9H228 13/20 0.53
S1PR4 O95977 4/20 0.53
MAP4K4 O95819 1/20 0.48
MINK1 Q8N4C8 1/20 0.48
S1PR3 Q99500 4/20 0.44
LTK P29376 1/20 0.42
TAOK1 Q7L7X3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9108025 0.86 S1PR1 (0.58) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL9107617 0.79 S1PR1 (0.58) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL9109266 0.79 S1PR1 (0.55) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL9111175 0.78 S1PR1 (0.60) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL16341310 0.78 S1PR1 (0.48) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL27942984 0.71 S1PR1 (0.54) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL27938162 0.70 S1PR1 (0.51) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL13415796 0.70 S1PR1 (1.00) S1PR1S1PR5S1PR4MAP4K4MINK1
SCHEMBL3043605 0.70 S1PR5 (1.00) S1PR1S1PR5S1PR4S1PR3
SCHEMBL9110235 0.69 S1PR1 (0.54) S1PR1S1PR5S1PR4MAP4K4MINK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646023-B1 NOVEL AZETIDINE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTOR MODULATORS ALLERGAN INC (US) 2015-01-07 EP claimed