SCHEMBL16360405

SCHEMBL16360405

CCCCCCNc1ncc2c(n1)-c1ccccc1C(c1ccc(/N=C/N(C)C)cc1)C2

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 4/20 0.41
FGFR2 P21802 2/20 0.41
CSF1R P07333 1/20 0.36
FGFR3 P22607 1/20 0.36
MERTK Q12866 13/20 0.35
TYRO3 Q06418 11/20 0.35
FLT3 P36888 8/20 0.35
GAS6 Q14393 8/20 0.35
AXL P30530 7/20 0.35
DNM2 P50570 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2489018 0.93 FGFR1 (0.41) FGFR1FGFR2CSF1RFGFR3MERTK
SCHEMBL2802907 0.93 FGFR1 (0.41) FGFR1FGFR2CSF1RFGFR3MERTK
SCHEMBL2489019 0.93 FGFR1 (0.41) FGFR1FGFR2CSF1RFGFR3MERTK
SCHEMBL2513190 0.89 FGFR1 (0.40) FGFR1FGFR2FGFR3
SCHEMBL2513192 0.89 FGFR1 (0.40) FGFR1FGFR2FGFR3
SCHEMBL2807869 0.84 FGFR1 (0.41) FGFR1FGFR2CSF1RFGFR3FLT3
SCHEMBL2807870 0.84 FGFR1 (0.41) FGFR1FGFR2CSF1RFGFR3FLT3
SCHEMBL14644885 0.84 FGFR1 (0.41) FGFR1FGFR2CSF1RFGFR3FLT3
SCHEMBL2803900 0.79 FGFR1 (0.54) FGFR1FGFR2CSF1RFGFR3MERTK
SCHEMBL2808949 0.78 FGFR1 (0.49) FGFR1FGFR2CSF1RFGFR3MERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379506-B1 SUBSTITUTED 5,6-DIHYDRO-6-PHENYLBENZO[F]ISOQUINOLIN-2-AMINE COMPOUNDS ARQULE INC (US) 2015-09-02 EP disclosed
WO-2010078421-A1 SUBSTITUTED 5,6-DIHYDRO-6-PHENYLBENZO[F] ISOQUINOLIN-2-AMINE COMPOUNDS ARQULE, INC. (US) 2010-07-08 WO disclosed