SCHEMBL16369452

SCHEMBL16369452

CC(C)Cn1c(=O)n(C)c(=O)c2c(Nc3ccccc3)n(Cc3ccc(-c4ncccn4)cc3)cc21

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 8/20 0.52
PDE1A P54750 7/20 0.52
PDE1C Q14123 7/20 0.52
PDE2A O00408 5/20 0.52
MAPT P10636 5/20 0.40
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
TP53 P04637 1/20 0.40
PKM P14618 1/20 0.39
SLC16A1 P53985 2/20 0.39
BRD4 O60885 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2462950 0.91 PDE1B (0.50) PDE1BPDE1APDE1CPDE2AMAPT
SCHEMBL9608325 0.90 PDE1A (0.41) PDE1BPDE1APDE1CPDE2ABRD4
SCHEMBL2454720 0.90 PDE1B (0.50) PDE1BPDE1APDE1CPDE2AMAPT
SCHEMBL9608334 0.87 PDE1B (0.52) PDE1BPDE1APDE1CPDE2AMAPT
SCHEMBL2458078 0.85 PDE1B (0.45) PDE1BPDE1APDE1CPDE2AMAPT
SCHEMBL2461370 0.85 PDE1A (0.49) PDE1BPDE1APDE1CPDE2AMAPT
SCHEMBL2454858 0.84 PDE1A (0.48) PDE1BPDE1APDE1CPDE2ASLC16A1
SCHEMBL2455942 0.84 PDE1B (0.48) PDE1BPDE1APDE1CPDE2AMAPT
SCHEMBL9609218 0.84 PDE1B (0.48) PDE1BPDE1APDE1CPDE2AMAPT
SCHEMBL9608337 0.84 PDE1B (0.48) PDE1BPDE1APDE1CPDE2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8927556-B2 1H-pyrrolo[3,4-D]pyrimidin-2(6H)-one compounds INTRA-CELLULAR THERAPIES, INC. (US) 2015-01-06 US disclosed
US-8927556-B2 1H-pyrrolo[3,4-D]pyrimidin-2(6H)-one compounds INTRA-CELLULAR THERAPIES, INC. (US) 2015-01-06 US disclosed