SCHEMBL16375982

SCHEMBL16375982

O=C(c1cc2ccccc2[nH]1)c1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 1.00
ERBB2 P04626 1/20 0.53
RET P07949 1/20 0.53
ERBB4 Q15303 1/20 0.53
HDAC3 O15379 3/20 0.50
HDAC1 Q13547 3/20 0.50
HDAC6 Q9UBN7 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5467893 0.80 EGFR (0.70) EGFRERBB2RETERBB4HDAC3
SCHEMBL5465521 0.72 EGFR (0.71) EGFRERBB2RETERBB4HDAC3
SCHEMBL5466827 0.72 EGFR (0.59) EGFRERBB2RETERBB4
SCHEMBL5469496 0.71 EGFR (0.65) EGFRERBB2RETERBB4HDAC3
SCHEMBL4740837 0.71 EGFR (0.74) EGFRERBB2RETERBB4HDAC3
SCHEMBL5464067 0.70 EGFR (0.68) EGFRERBB2RETERBB4HDAC3
SCHEMBL5465513 0.70 EGFR (0.60) EGFRERBB2RETERBB4HDAC3
SCHEMBL5462878 0.70 EGFR (0.58) EGFRERBB2RETERBB4HDAC3
SCHEMBL5469233 0.70 EGFR (0.60) EGFRERBB2RETERBB4
SCHEMBL5465619 0.70 EGFR (0.63) EGFRERBB2RETERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015000959-A1 4-AMINO-6-ARYL[2,3-D]PYRIMIDINES FOR THE INHIBITION OF EGFR TYROSINE KINASE NORWEGIAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (NTNU) (NO) 2015-01-08 WO disclosed