SCHEMBL16376342

SCHEMBL16376342

Cn1ccc2c(-c3ncc(F)c(N4CCC[C@@H]4C(=O)NCC(F)(F)F)n3)ccnc21

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GUCY1B2 O75343 3/20 0.38
GUCY1A2 P33402 3/20 0.38
GUCY1A1 Q02108 3/20 0.38
GUCY1B1 Q02153 3/20 0.38
AADAT Q8N5Z0 13/20 0.36
CAMKK1 Q8N5S9 1/20 0.35
CAMKK2 Q96RR4 1/20 0.35
JAK3 P52333 2/20 0.35
JAK2 O60674 1/20 0.35
ACACB O00763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16376343 1.00 GUCY1B2 (0.38) GUCY1B2GUCY1A2GUCY1A1GUCY1B1AADAT
SCHEMBL14494146 0.85 JAK1 (0.44) GUCY1B2GUCY1A2GUCY1A1GUCY1B1JAK3
SCHEMBL14494151 0.85 JAK1 (0.44) GUCY1B2GUCY1A2GUCY1A1GUCY1B1JAK3
SCHEMBL10044624 0.81 GUCY1B2 (0.40) GUCY1B2GUCY1A2GUCY1A1GUCY1B1AADAT
SCHEMBL10044611 0.81 GUCY1B2 (0.40) GUCY1B2GUCY1A2GUCY1A1GUCY1B1AADAT
SCHEMBL2630353 0.79 JAK3 (0.55) GUCY1B2GUCY1A2GUCY1A1GUCY1B1JAK3
SCHEMBL2630352 0.79 JAK3 (0.55) GUCY1B2GUCY1A2GUCY1A1GUCY1B1JAK3
SCHEMBL13305968 0.79 GUCY1B2 (0.40) GUCY1B2GUCY1A2GUCY1A1GUCY1B1AADAT
SCHEMBL10044597 0.78 F2 (0.41) GUCY1B2GUCY1A2GUCY1A1GUCY1B1AADAT
SCHEMBL10044617 0.78 F2 (0.41) GUCY1B2GUCY1A2GUCY1A1GUCY1B1AADAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921376-B2 Pyrrolopyridines useful as inhibitors of protein kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-12-30 US disclosed