SCHEMBL16404607

SCHEMBL16404607

Cc1noc(C)c1-c1ccc(F)cc1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.66
BRD2 P25440 1/20 0.66
MLYCD O95822 1/20 0.58
GPR55 Q9Y2T6 1/20 0.56
PTGS2 P35354 3/20 0.54
PTGS1 P23219 1/20 0.54
LMNA P02545 3/20 0.52
CYP1A2 P05177 3/20 0.52
CYP3A4 P08684 3/20 0.52
CYP2C19 P33261 3/20 0.52
CLK4 Q9HAZ1 2/20 0.52
USP2 O75604 1/20 0.52
TP53 P04637 1/20 0.52
CYP2D6 P10635 1/20 0.52
HIF1A Q16665 1/20 0.52
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
PIK3CD O00329 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300240 0.83 BRD4 (0.70) BRD4BRD2MLYCD
SCHEMBL17532580 0.81 BRD4 (0.68) BRD4BRD2GPR55PTGS2PTGS1
SCHEMBL14678367 0.80 BRD4 (0.66) BRD4BRD2MLYCDLMNACYP3A4
SCHEMBL12077969 0.80 BRD4 (0.55) BRD4BRD2MLYCDLMNA
SCHEMBL1772573 0.80 BRD4 (0.66) BRD4BRD2MLYCDLMNACYP1A2
SCHEMBL3885694 0.80 BRD4 (0.66) BRD4BRD2MLYCD
SCHEMBL12362813 0.80 BRD4 (0.66) BRD4BRD2MLYCD
3,5-Dimethyl-4-Phenylisoxazole SCHEMBL12134072 0.79 BRD4 (1.00) BRD4BRD2MLYCDPTGS2PTGS1
Hydrochloric Acid SCHEMBL23174957 0.78 BRD4 (0.63) BRD4BRD2MLYCD
SCHEMBL3818394 0.78 BRD4 (0.49) BRD4BRD2MLYCDGPR55PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429993-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BOEHRINGER INGELHEIM INT (DE) 2015-01-21 EP disclosed