Aspartic Acid

Aspartic Acid

SCHEMBL16431397

N[C@@H](CC(=O)[O-])C(=O)[O-].N[C@@H](CC(=O)[O-])C(=O)[O-].[Pb+4]

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC6A2SLC6A3SSTR1SSTR2SSTR3SSTR5

The experimentally established mechanism targets of Aspartic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA4 P22748 4/20 0.48
CTSL P07711 1/20 0.44
CPT2 P23786 1/20 0.43
CPT1A P50416 1/20 0.43
CA2 P00918 1/20 0.42
SLC22A16 Q86VW1 1/20 0.36
GRIK1 P39086 1/20 0.31
GRIK2 Q13002 1/20 0.31
GRM1 Q13255 1/20 0.31
GRM2 Q14416 1/20 0.31
GSR P00390 1/20 0.31
PTGS1 P23219 1/20 0.31
SLC7A11 Q9UPY5 1/20 0.31
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aspartic Acid SCHEMBL18130875 1.00 CA4 (0.48) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL20400343 0.94 CA4 (0.48) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL120390 0.94 CA4 (0.52) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL11903451 0.94 CA4 (0.48) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL1655126 0.94 CA4 (0.48) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL11903448 0.94 CA4 (0.48) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL7635443 0.94 CA4 (0.48) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL21054602 0.94 CA4 (0.52) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL22401093 0.94 CA4 (0.52) CA4CTSLCPT2CPT1ACA2
Aspartic Acid SCHEMBL161238 0.94 CA4 (0.48) CA4CTSLCPT2CPT1ACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250090463-A1 INHALED IMATINIB FOR TREATMENT OF PULMONARY ARTERIAL HYPERTENSION (PAH) AVALYN PHARMA INC. 2025-03-20 US disclosed
EP-3027026-B1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF AVALYN PHARMA INC (US) 2024-11-13 EP disclosed
US-11980689-B2 Inhaled imatinib for treatment of pulmonary arterial hypertension (PAH) AVALYN PHARMA INC. (US) 2024-05-14 US disclosed
US-20220087937-A1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF AVALYN PHARMA INC. 2022-03-24 US disclosed
US-20210093570-A1 INHALED IMATINIB FOR TREATMENT OF PULMONARY ARTERIAL HYPERTENSION (PAH) AVALYN PHARMA INC. 2021-04-01 US disclosed
US-20210093569-A1 INHALED IMATINIB FOR TREATMENT OF PULMONARY ARTERIAL HYPERTENSION (PAH) AVALYN PHARMA INC. 2021-04-01 US disclosed
EP-3782604-A1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF Windward Pharma, Inc. (US) 2021-02-24 EP disclosed
EP-3027026-A1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF Windward Pharma, Inc. (US) 2016-06-08 EP disclosed
US-20150044288-A1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF AVALYN PHARMA INC. 2015-02-12 US disclosed
WO-2015017728-A1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF WINDWARD PHARMA, INC. (US) 2015-02-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210093569-A1 INHALED IMATINIB FOR TREATMENT OF PULMONARY ARTERIAL HYPERTENSION (PAH) ALK, JAK1, PAH CA4 1016/4885CTSL 4751/4885CPT2 4221/4885
US-20150044288-A1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF ALK, JAK1, ABL1 CA4 1930/4885CTSL 4654/4885CPT2 4558/4885
US-20250090463-A1 INHALED IMATINIB FOR TREATMENT OF PULMONARY ARTERIAL HYPERTENSION (PAH) ALK, JAK1, PAH CA4 1016/4885CTSL 4751/4885CPT2 4221/4885
US-20210093570-A1 INHALED IMATINIB FOR TREATMENT OF PULMONARY ARTERIAL HYPERTENSION (PAH) ALK, JAK1, PAH CA4 1016/4885CTSL 4751/4885CPT2 4221/4885
US-20220087937-A1 AEROSOL TYROSINE KINASE INHIBITOR COMPOUNDS AND USES THEREOF ALK, JAK1, ABL1 CA4 1930/4885CTSL 4654/4885CPT2 4558/4885
US-11980689-B2 Inhaled imatinib for treatment of pulmonary arterial hypertension (PAH) ALK, JAK1, PAH CA4 1016/4885CTSL 4751/4885CPT2 4221/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.