SCHEMBL16455012

SCHEMBL16455012

Brc1ccc2c(c1)-c1ccccc1Oc1ccccc1-c1cc(Br)ccc1O2

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.65
MAPK1 P28482 3/20 0.45
KDM4E B2RXH2 1/20 0.45
ATM Q13315 1/20 0.45
PTPRC P08575 1/20 0.45
SIRT1 Q96EB6 1/20 0.43
CYP19A1 P11511 1/20 0.39
CYP1A2 P05177 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HTR2A P28223 4/20 0.38
HTR2C P28335 4/20 0.38
DRD2 P14416 2/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2C P18825 1/20 0.38
DRD1 P21728 1/20 0.38
HTR7 P34969 1/20 0.38
HRH1 P35367 1/20 0.38
DRD3 P35462 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16800898 0.98 AHR (0.63) AHRMAPK1KDM4EATMPTPRC
SCHEMBL16800942 0.93 AHR (0.61) AHRMAPK1KDM4EATMPTPRC
SCHEMBL19885489 0.89 AHR (0.57) AHRMAPK1KDM4EATMPTPRC
SCHEMBL10956695 0.84 AHR (0.57) AHRMAPK1KDM4EATMPTPRC
SCHEMBL18159686 0.83 AHR (0.50) AHRMAPK1PTPRCSIRT1CYP19A1
SCHEMBL17283693 0.81 MAPK1 (0.65) AHRMAPK1KDM4EATMPTPRC
SCHEMBL10952987 0.81 AHR (0.53) AHRMAPK1KDM4EATMPTPRC
SCHEMBL47076 0.79 AHR (1.00) AHRSIRT1HTR2AHTR2CDRD2
SCHEMBL30434673 0.79 AHR (1.00) AHRSIRT1HTR2AHTR2CDRD2
SCHEMBL10952178 0.79 AHR (0.50) AHRMAPK1KDM4EATMPTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9425401-B2 9,9′-spirobixanthene derivatives for electroluminescent devices MERCK PATENT GMBH (DE) 2016-08-23 US disclosed
US-20150045529-A1 9,9'-SPIROBIXANTHENE DERIVATIVES FOR ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2015-02-12 US disclosed