SCHEMBL1646288

SCHEMBL1646288

Fc1cccc(F)c1-c1c(-c2ccncc2)cnn1C1CCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 11/20 0.47
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
RAB9A P51151 1/20 0.39
GRM2 Q14416 1/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647081 0.97 S1PR1 (0.50) S1PR1NPC1LMNARAB9AGRM2
SCHEMBL1554460 0.73 NPC1 (0.39) S1PR1NPC1LMNARAB9AHDAC9
SCHEMBL1645859 0.72 CHRM1 (0.47) LMNA
SCHEMBL1645694 0.72 BRAF (0.45) NPC1LMNARAB9A
SCHEMBL6077431 0.71 MAPK14 (0.52) S1PR1PTGS1PTGS2
SCHEMBL1648133 0.70 S1PR1 (0.40) S1PR1NPC1LMNARAB9AGRM2
SCHEMBL1646195 0.70 S1PR1 (0.52) S1PR1NPC1LMNARAB9AALDH1A1
SCHEMBL1646250 0.69 BRAF (0.47) NPC1LMNARAB9A
SCHEMBL1646948 0.69 RIPK3 (0.36) S1PR1NPC1LMNARAB9AALDH1A1
SCHEMBL771248 0.68 S1PR1 (0.94) S1PR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed