SCHEMBL16472008

SCHEMBL16472008

CC(=O)c1ccc2c(c1)CC1(C2)C(=O)Nc2ncccc21

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADM2 Q7Z4H4 9/20 0.52
CALCRL Q16602 11/20 0.51
CALCB P10092 8/20 0.51
RAMP1 O60894 4/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1815456 0.89 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL29996226 0.89 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL7030609 0.89 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL13376816 0.88 CALCRL (0.49) ADM2CALCRLCALCBRAMP1
SCHEMBL31084970 0.87 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL15236128 0.87 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL12655038 0.87 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL22796626 0.87 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL29416274 0.87 CALCRL (0.51) ADM2CALCRLCALCBRAMP1
SCHEMBL29517886 0.87 CALCRL (0.51) ADM2CALCRLCALCBRAMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912653-B1 HETEROCYCLIC BENZODIAZEPINE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2014-01-01 EP disclosed