SCHEMBL16474146

SCHEMBL16474146

CCC(C)C(C(=O)OC(C)(C)I)c1ccc(CN2N=C(c3ccccc3)OCC2=O)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
CHRM5 P08912 1/20 0.33
CYP2D6 P10635 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
KMT2A Q03164 1/20 0.32
MAOB P27338 2/20 0.32
ALDH1A1 P00352 2/20 0.31
GAA P10253 1/20 0.31
THRB P10828 1/20 0.31
POLB P06746 1/20 0.31
HTT P42858 1/20 0.31
PGR P06401 1/20 0.31
TSHR P16473 1/20 0.30
PKM P14618 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517218 0.93 CHRM2 (0.34) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL517151 0.86 KMT2A (0.37) CYP2D6KMT2AMAOBALDH1A1GAA
SCHEMBL3703386 0.86 KMT2A (0.32) KMT2AMAOBALDH1A1GAATHRB
SCHEMBL3691213 0.85 MAOB (0.35) KMT2AMAOBALDH1A1GAATHRB
SCHEMBL3691767 0.85 KMT2A (0.32) CYP2D6KMT2AMAOBALDH1A1GAA
SCHEMBL1178303 0.84 KMT2A (0.34) CYP2D6KMT2AMAOBALDH1A1GAA
SCHEMBL7603996 0.84 KMT2A (0.36) CYP2D6KMT2AMAOBALDH1A1GAA
SCHEMBL3700165 0.83 KMT2A (0.39) KMT2AMAOBALDH1A1GAAHTT
SCHEMBL16474230 0.82 AAK1 (0.32) KMT2AMAOBALDH1A1GAATHRB
SCHEMBL1177873 0.80 KMT2A (0.39) CYP2D6KMT2AMAOBALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406215-B1 OXO-HETEROCYCLICALLY SUBSTITUTED ALKYL CARBOXYLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2014-04-16 EP disclosed