SCHEMBL16478299

SCHEMBL16478299

COCCCn1c(=O)oc2ccc(-c3ccc(CC(NC(=O)C4(NC(=O)O)CCCC4)C(N)=O)cc3)cc21

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSC P53634 4/20 0.50
ITGB1 P05556 6/20 0.39
ITGA4 P13612 6/20 0.39
ITGB7 P26010 5/20 0.39
TACR2 P21452 2/20 0.39
ASAH1 Q13510 1/20 0.39
ECE1 P42892 2/20 0.38
NPPA P01160 1/20 0.38
MME P08473 1/20 0.38
KCNH2 Q12809 1/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
TSHR P16473 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299037 0.94 CTSC (0.49) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL16478309 0.91 CTSC (0.47) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL16478310 0.91 CTSC (0.47) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL299685 0.90 CTSC (0.49) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL16478294 0.87 CTSC (0.45) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL16478321 0.86 CTSC (0.45) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL7867141 0.85 CTSC (0.47) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL9888335 0.85 CTSC (0.46) CTSCITGB1ITGA4ITGB7TACR2
SCHEMBL2885392 0.82 CTSC (0.62) CTSCKCNH2
SCHEMBL7873698 0.81 CTSC (0.46) CTSCITGB1ITGA4ITGB7TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011154677-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL] 1-AMINOCYCLOALK-1-YLCARBOXAMIDE COMPOUNDS - 760 ASTRAZENECA AB (SE) 2011-12-15 WO disclosed