SCHEMBL16480397

SCHEMBL16480397

CC1CCC(=O)N1c1ccc(C#N)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.43
ABL1 P00519 2/20 0.40
CHRM2 P08172 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
PARP1 P09874 3/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13934938 0.84 AR (0.62) ARSLC6A2SLC6A4SLC6A3
SCHEMBL13934721 0.83 AR (0.57) AR
SCHEMBL9891769 0.83 AR (0.40) AR
SCHEMBL9892990 0.83 ABL1 (0.44) ABL1PARP1SLC6A2SLC6A4SLC6A3
SCHEMBL19745913 0.83 AR (0.38) ARPARP1
SCHEMBL19745911 0.83 AR (0.38) ARPARP1
SCHEMBL9103503 0.81 NR3C2 (0.40) ARCHRM2CHRM5CHRM1
SCHEMBL19745517 0.81 HDAC1 (0.52) ARPARP1
SCHEMBL9103496 0.81 NR3C2 (0.40) ARCHRM2CHRM5CHRM1
SCHEMBL19745519 0.81 HDAC1 (0.52) ARPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8629157-B2 Pyrrolidine compounds which modulate the CB2 receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-14 US disclosed