SCHEMBL16485802

SCHEMBL16485802

CC(C)N1Cc2cc(-c3ccc(C[C@H](NC(=O)C4(NC(=O)OC(C)(C)C)CCCCC4)C(N)=O)cc3)cnc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 12/20 0.38
ITGA4 P13612 2/20 0.35
ITGB7 P26010 2/20 0.35
RET P07949 2/20 0.34
REN P00797 1/20 0.34
APC P25054 1/20 0.33
LCK P06239 1/20 0.33
GRB2 P62993 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2893127 0.91 ECE1 (0.38) ECE1ITGA4ITGB7RETREN
SCHEMBL2893129 0.91 ECE1 (0.38) ECE1ITGA4ITGB7RETREN
SCHEMBL16478298 0.90 ECE1 (0.43) ECE1ITGA4
SCHEMBL16485829 0.88 CTSC (0.40) RETCTSK
SCHEMBL16485757 0.85 ECE1 (0.40) ECE1ITGA4ITGB7RETREN
SCHEMBL9886055 0.84 CTSC (0.41) ECE1ITGA4ITGB7RETREN
SCHEMBL16478325 0.81 ECE1 (0.42) ECE1ITGA4ITGB7CTSK
SCHEMBL16485763 0.80 ECE1 (0.41) ECE1ITGA4ITGB7RENAPC
SCHEMBL16485782 0.79 CTSC (0.48) RETCTSSCTSK
SCHEMBL16485771 0.79 CTSC (0.38) ECE1ITGA4ITGB7RENAPC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011154677-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL] 1-AMINOCYCLOALK-1-YLCARBOXAMIDE COMPOUNDS - 760 ASTRAZENECA AB (SE) 2011-12-15 WO disclosed