SCHEMBL16487606

SCHEMBL16487606

O=C1CCc2cc(S(=O)(=O)NC(Cc3ccccc3)C(=O)N3CCCC3)ccc2N1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2D6 P10635 1/20 0.70
KMT2A Q03164 1/20 0.70
THRB P10828 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
OGT O15294 8/20 0.66
MAPT P10636 4/20 0.66
TP53 P04637 1/20 0.66
LMNA P02545 1/20 0.65
TSHR P16473 1/20 0.65
ALDH1A1 P00352 4/20 0.63
MAPK1 P28482 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16487680 0.99 MEN1 (0.69) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487593 0.99 MEN1 (0.69) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487691 0.93 MEN1 (0.70) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487682 0.92 MEN1 (0.67) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487684 0.91 MEN1 (0.68) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487697 0.91 OGT (0.68) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487614 0.90 KMT2A (0.65) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487634 0.90 OGT (0.68) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487626 0.90 MEN1 (0.62) MEN1CYP3A4CYP2D6KMT2ATHRB
SCHEMBL16487699 0.90 OGT (0.77) MEN1CYP3A4CYP2D6KMT2ATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8957075-B2 O-GlcNAc transferase inhibitors and uses thereof PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-02-17 US disclosed
US-8957075-B2 O-GlcNAc transferase inhibitors and uses thereof PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-02-17 US disclosed