SCHEMBL16489072

SCHEMBL16489072

CCN1CCN(C(=O)c2cccc(-c3cncc(C(=O)Nc4ccccc4)n3)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATR Q13535 11/20 0.56
PRKAA2 P54646 2/20 0.50
SCN2A Q99250 2/20 0.46
SCN10A Q9Y5Y9 2/20 0.46
CCNC P24863 2/20 0.46
CDK8 P49336 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16420791 0.93 ATR (0.57) ATRPRKAA2SCN2ASCN10ACCNC
SCHEMBL16420777 0.89 ATR (0.69) ATRSCN2ASCN10ACCNCCDK8
SCHEMBL16420775 0.88 ATR (0.67) ATRCCNCCDK8MEN1KMT2A
SCHEMBL19101115 0.87 ATR (0.66) ATRCCNCCDK8MEN1KMT2A
SCHEMBL16489089 0.87 ATR (0.72) ATRPRKAA2SCN2ASCN10ACCNC
SCHEMBL19101135 0.87 ATR (0.61) ATRPRKAA2CCNCCDK8MEN1
SCHEMBL16420790 0.85 ATR (0.69) ATRCCNCCDK8
SCHEMBL16489060 0.85 ATR (0.69) ATRMEN1KMT2A
SCHEMBL19101118 0.85 ATR (0.54) ATRSCN2ASCN10A
SCHEMBL16420769 0.84 ATR (0.71) ATRPRKAA2SCN2ASCN10ACCNC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150051187-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED 2015-02-19 US disclosed
US-20150030539-A1 COMPOUNDS FOR USE IN IMAGING, DIAGNOSING AND/OR TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM OR OF TUMORS PIRAMAL IMAGING SA (CH) 2015-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150030539-A1 COMPOUNDS FOR USE IN IMAGING, DIAGNOSING AND/OR TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM OR OF TUMORS PMP22, MEN1, VHL ATR 2406/4885PRKAA2 4246/4885SCN2A 1805/4885
US-20150051187-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK1, MAP3K5 ATR 1/4885PRKAA2 98/4885SCN2A 2823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.