SCHEMBL16489083

SCHEMBL16489083

CCc1ccc(-c2nnc(-c3nc(-c4ccc(S(=O)(=O)CC)cc4)cnc3N)o2)cc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATR Q13535 19/20 0.62
GSK3B P49841 1/20 0.62
PRKDC P78527 1/20 0.62
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2483511 0.90 ATR (0.76) ATRGSK3BPRKDC
SCHEMBL2482117 0.90 ATR (0.66) ATRGSK3BPRKDCKCNH2
SCHEMBL20283870 0.89 ATR (0.80) ATRGSK3BPRKDC
SCHEMBL16070049 0.83 ATR (0.63) ATRGSK3BPRKDCKCNH2
SCHEMBL3048753 0.82 ATR (0.67) ATRGSK3BPRKDC
SCHEMBL16093104 0.81 ATR (0.58) ATRGSK3BPRKDC
SCHEMBL13345797 0.81 ATR (0.79) ATRPRKDCKCNH2
SCHEMBL13138284 0.81 ATR (0.67) ATRGSK3BPRKDCKCNH2
SCHEMBL2484306 0.81 ATR (0.80) ATRGSK3BPRKDC
SCHEMBL24248210 0.80 ATR (0.71) ATRGSK3BPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150051187-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED 2015-02-19 US disclosed
US-20150030539-A1 COMPOUNDS FOR USE IN IMAGING, DIAGNOSING AND/OR TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM OR OF TUMORS PIRAMAL IMAGING SA (CH) 2015-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150030539-A1 COMPOUNDS FOR USE IN IMAGING, DIAGNOSING AND/OR TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM OR OF TUMORS PMP22, MEN1, VHL ATR 2406/4885GSK3B 1449/4885PRKDC 4071/4885
US-20150051187-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK1, MAP3K5 ATR 1/4885GSK3B 216/4885PRKDC 23/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.