SCHEMBL16495205

SCHEMBL16495205

NCc1cc2c(Nc3ncc(Cc4ccc5[nH]ccc5c4)c(N)n3)cccc2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.35
EGFR P00533 2/20 0.35
PDGFRB P09619 1/20 0.35
ULK1 O75385 1/20 0.33
DHFR P00374 2/20 0.33
PLK2 Q9NYY3 1/20 0.33
FLT1 P17948 1/20 0.33
CDK1 P06493 2/20 0.32
LOXL2 Q9Y4K0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16494735 0.91 KDR (0.34) KDREGFRPDGFRBULK1DHFR
SCHEMBL16494704 0.90 KDR (0.37) KDREGFRPDGFRBULK1DHFR
SCHEMBL16495033 0.88 SYK (0.39) ULK1DHFRPLK2
SCHEMBL2598786 0.88 PLK2 (0.41) KDRULK1DHFRPLK2CDK1
SCHEMBL2598707 0.86 EPHB4 (0.42)
SCHEMBL16494296 0.86 SYK (0.40) KDREGFRPDGFRBULK1DHFR
SCHEMBL16495173 0.81 EGFR (0.35) KDREGFRULK1DHFRFLT1
SCHEMBL2598631 0.80 PIK3CA (0.42) DHFRPLK2
SCHEMBL2598767 0.80 SYK (0.41) PLK2
SCHEMBL16494266 0.80 HTR2A (0.37) KDRULK1DHFRCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2395001-A1 Novel pyrimidine derivatives Chemilia AB (SE) 2011-12-14 EP disclosed