SCHEMBL16497950

SCHEMBL16497950

O=C(NC1CC[C@H]2CN(Cc3ccccc3)CC12)C(C1CCCCC1)C1CCCCC1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 4/20 0.74
KCNH2 Q12809 2/20 0.74
ALDH1A1 P00352 1/20 0.45
DPP7 Q9UHL4 1/20 0.43
CNR1 P21554 2/20 0.43
CNR2 P34972 2/20 0.43
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
KMT2A Q03164 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
SCN9A Q15858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65348 1.00 CACNA1B (0.74) CACNA1BKCNH2ALDH1A1DPP7CNR1
SCHEMBL66978 1.00 CACNA1B (0.74) CACNA1BKCNH2ALDH1A1DPP7CNR1
SCHEMBL2840316 1.00 CACNA1B (0.74) CACNA1BKCNH2ALDH1A1DPP7CNR1
SCHEMBL66676 1.00 CACNA1B (0.74) CACNA1BKCNH2ALDH1A1DPP7CNR1
SCHEMBL16497968 1.00 CACNA1B (0.74) CACNA1BKCNH2ALDH1A1DPP7CNR1
SCHEMBL2844033 0.89 KCNH2 (0.61) CACNA1BKCNH2ALDH1A1CYP2C19SMN1; SMN2
SCHEMBL2844031 0.89 KCNH2 (0.61) CACNA1BKCNH2ALDH1A1CYP2C19SMN1; SMN2
SCHEMBL65548 0.89 KCNH2 (0.61) CACNA1BKCNH2ALDH1A1CYP2C19SMN1; SMN2
SCHEMBL2849638 0.89 KCNH2 (0.61) CACNA1BKCNH2ALDH1A1CYP2C19SMN1; SMN2
SCHEMBL65848 0.89 KCNH2 (0.61) CACNA1BKCNH2ALDH1A1CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149995-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA [C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2011-12-01 WO claimed
WO-2011149995-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA [C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2011-12-01 WO disclosed