SCHEMBL16497983

SCHEMBL16497983

CC(C)C(C(=O)NC1CCC2CN(Cc3cccc(Cl)c3)CC21)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.53
KCNH2 Q12809 2/20 0.51
ACKR3 P25106 1/20 0.46
SIGMAR1 Q99720 2/20 0.44
FAAH O00519 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 2/20 0.41
HTT P42858 2/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CCR5 P51681 1/20 0.40
DRD4 P21917 2/20 0.40
HTR4 Q13639 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL67438 1.00 CACNA1B (0.53) CACNA1BKCNH2ACKR3SIGMAR1FAAH
SCHEMBL65881 0.92 CACNA1B (0.52) CACNA1BKCNH2ACKR3MEN1KMT2A
SCHEMBL16497753 0.92 CACNA1B (0.52) CACNA1BKCNH2ACKR3MEN1KMT2A
SCHEMBL2842532 0.92 CACNA1B (0.52) CACNA1BKCNH2ACKR3MEN1KMT2A
SCHEMBL2842533 0.92 CACNA1B (0.52) CACNA1BKCNH2ACKR3MEN1KMT2A
SCHEMBL67094 0.92 CACNA1B (0.52) CACNA1BKCNH2ACKR3MEN1KMT2A
SCHEMBL67560 0.92 CACNA1B (0.52) CACNA1BKCNH2ACKR3MEN1KMT2A
SCHEMBL67382 0.91 CACNA1B (0.49) CACNA1BKCNH2ACKR3SIGMAR1MEN1
SCHEMBL16497798 0.91 CACNA1B (0.49) CACNA1BKCNH2ACKR3SIGMAR1MEN1
SCHEMBL65591 0.90 CACNA1B (0.53) CACNA1BKCNH2ACKR3FAAHMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149995-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA [C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2011-12-01 WO claimed
WO-2011149995-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA [C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2011-12-01 WO disclosed