SCHEMBL16498121

SCHEMBL16498121

O=C(O)c1cc(F)cnc1OCc1ccccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
TP53 P04637 1/20 0.49
HTT P42858 1/20 0.49
MCL1 Q07820 1/20 0.47
MRGPRX4 Q96LA9 3/20 0.45
ALKBH1 Q13686 1/20 0.44
SGMS2 Q8NHU3 2/20 0.43
GCK P35557 1/20 0.43
FABP4 P15090 1/20 0.42
FABP5 Q01469 1/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012447 0.87 MCL1 (0.52) NR4A2NPC1RAB9ATP53HTT
SCHEMBL16498112 0.84 PARP10 (0.51) TP53HTTALKBH1MEN1KMT2A
SCHEMBL16498677 0.82 LRRK2 (0.48) NR4A2MCL1MRGPRX4ALKBH1MEN1
SCHEMBL16498119 0.80 FFAR1 (0.42) HTTMRGPRX4SGMS2LRRK2
SCHEMBL2292252 0.79 TP53 (0.62) NR4A2NPC1RAB9ATP53HTT
SCHEMBL16498161 0.78 SYK (0.44) NPC1RAB9AKMT2A
SCHEMBL16498273 0.77 NAPRT (0.39) LRRK2
SCHEMBL16498100 0.75 GRM4 (0.52) SGMS2MEN1KMT2ALRRK2
SCHEMBL16498135 0.75 GRM4 (0.49) NR4A2MEN1KMT2ALRRK2
SCHEMBL16498549 0.73 NAPRT (0.40) MRGPRX4LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151651-A1 BENZODIAZEPINE COMPOUNDS USEFUL FOR THE TREATMENT OF HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2011-12-08 WO disclosed