SCHEMBL16504334

SCHEMBL16504334

CC(C)[Si](OCCSc1ccccc1-c1nnc2ccc(O[C@H]3CC[C@H](N)c4ccccc43)cn12)(C(C)C)C(C)C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.34
SLC6A3 Q01959 2/20 0.34
SLC6A4 P31645 1/20 0.34
MAPK14 Q16539 15/20 0.34
MAPK12 P53778 3/20 0.33
MAPK11 Q15759 3/20 0.33
MAPK13 O15264 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15028559 1.00 SLC6A2 (0.34) SLC6A2SLC6A3SLC6A4MAPK14MAPK12
SCHEMBL16504331 1.00 SLC6A2 (0.34) SLC6A2SLC6A3SLC6A4MAPK14MAPK12
SCHEMBL14990398 0.82 MAPK14 (0.32) SLC6A2SLC6A3SLC6A4MAPK14MAPK12
SCHEMBL15007641 0.79 MAPK14 (0.37) SLC6A2SLC6A3SLC6A4MAPK14MAPK12
SCHEMBL15007640 0.79 MAPK14 (0.37) SLC6A2SLC6A3SLC6A4MAPK14MAPK12
SCHEMBL15007883 0.77 MAPK14 (0.41) MAPK14MAPK12MAPK11MAPK13
SCHEMBL15006725 0.76 SLC6A2 (0.41) SLC6A2SLC6A3SLC6A4MAPK14MAPK12
SCHEMBL15028544 0.76 MAPK14 (0.38) MAPK14
SCHEMBL981551 0.76 PIM1 (0.36) MAPK14MAPK11
SCHEMBL15008720 0.76 MAPK14 (0.44) MAPK14MAPK12MAPK11MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788345-B1 DERIVATIVES OF 4-HYDROXY-1,2,3,4-TETRAHYDRONAPHTALEN-1-YL UREA AND THEIR USE IN THE TREATMENT OF, INTER ALIA, DISEASES OF THE RESPIRATORY TRACT CHIESI FARM SPA (IT) 2020-06-10 EP disclosed
US-9458154-B2 Kinase inhibitors CHIESI FARMACEUTICI S.P.A. (IT) 2016-10-04 US disclosed
US-20150057273-A1 KINASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2015-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150057273-A1 KINASE INHIBITORS MAPK1, MAP3K1, MAPK4 SLC6A2 4577/4885SLC6A3 4458/4885SLC6A4 4366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.