SCHEMBL1654993

SCHEMBL1654993

O=C(Nc1cccc(CCCN2CCOCC2)c1C(F)(F)F)c1cccnc1NCc1ccncc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.56
KDR P35968 15/20 0.52
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
AURKA O14965 1/20 0.42
RPS6KB1 P23443 1/20 0.42
AURKB Q96GD4 1/20 0.42
TRPV4 Q9HBA0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL445762 0.82 KDR (0.68) ABCB1KDRTRPV4
SCHEMBL429577 0.80 ABCB1 (0.61) ABCB1KDR
SCHEMBL1654453 0.77 KDR (0.49) ABCB1KDR
SCHEMBL427599 0.74 ABCB1 (0.79) ABCB1KDRKDM4EMAPT
SCHEMBL427658 0.74 ABCB1 (0.69) ABCB1KDR
SCHEMBL446249 0.74 KDR (0.70) ABCB1KDRMAPT
SCHEMBL3106416 0.73 KDR (0.66) ABCB1KDR
SCHEMBL426633 0.72 ABCB1 (1.00) ABCB1KDRKDM4EMAPT
SCHEMBL3108804 0.72 KDR (0.65) ABCB1KDR
SCHEMBL427754 0.72 KDR (0.55) ABCB1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2311829-A1 Substituted alkylamine derivatives and methods of use Amgen Inc. (US) 2011-04-20 EP disclosed