SCHEMBL1655428

SCHEMBL1655428

O=C1CC=CC=C1c1ncncn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8939186 0.82
SCHEMBL5848037 0.76
SCHEMBL6643593 0.67
SCHEMBL13386056 0.66 NISCH (0.37)
SCHEMBL5704894 0.66 KDM4A (0.37)
SCHEMBL5138828 0.66 BRD4 (0.35)
SCHEMBL7395758 0.65
SCHEMBL9616686 0.65 CCR1 (0.48)
SCHEMBL4750813 0.64
SCHEMBL668518 0.64 BACE1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1722859-A1 A BASE COMPOSITION FOR PREPARING MULTI-FUNCTIONAL FORMULATIONS FOR CARE AND PROTECTION OF THE SKIN AND HAIR Natura Cosméticos S.A. (BR) 2006-11-22 EP claimed
WO-2005060923-A1 A BASE COMPOSITION FOR PREPARING MULTI-FUNCTIONAL FORMULATIONS FOR CARE AND PROTECTION OF THE SKIN AND HAIR Natura Cosméticos S.A. (BR) 2005-07-07 WO claimed
WO-2023046842-A1 USE OF WATER-SOLUBLE LIGNIN AS AN ANTI-UV FILTER CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2023-03-30 WO disclosed
CN-114042002-A Mild and full-green sun block capable of remarkably increasing SPF (specific pathogen free) and preparation method thereof 广东馨柯生命科学有限公司 2022-02-15 CN disclosed
WO-2020231163-A1 ULTRAVIOLET LIGHT BLOCKING COMPOSITION COMPRISING BIS-ETHYLHEXYLOXYPHENOL METHOXYPHENYL TRIAZINE COMPOSITE FORMULATION ㈜아모레퍼시픽 2020-11-19 WO disclosed
EP-3675808-A1 WATER BASED CONCENTRATED PRODUCT FORMS OF OIL-SOLUBLE ORGANIC UV ABSORBERS BASF SE (DE) 2020-07-08 EP disclosed
WO-2019042999-A1 WATER BASED CONCENTRATED PRODUCT FORMS OF OIL-SOLUBLE ORGANIC UV ABSORBERS BASF SE (DE) 2019-03-07 WO disclosed
EP-3229766-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2017-10-18 EP disclosed
EP-3227016-A1 MICROCAPSULES BASF SE (DE) 2017-10-11 EP disclosed
WO-2016091930-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2016-06-16 WO disclosed
US-8535648-B2 Stabilization of UV-sensitive active ingredients BASF SE (DE) 2013-09-17 US disclosed
WO-2011048011-A2 BENZOTROPOLONE DERIVATIVES AS ANTIMICROBIAL AGENTS BASF SE (DE) 2011-04-28 WO disclosed
US-20100104523-A1 STABILIZATION OF UV-SENSITIVE ACTIVE INGREDIENTS CIBA CORPORATION (US) 2010-04-29 US disclosed
EP-2059220-A1 SEMI-FINISHED PRODUCT IN THE MANUFACTURE OF A COMPOSITION FOR SKIN OR HAIR CARE Oy Granula AB LTD (FI) 2009-05-20 EP disclosed
WO-2008020112-A1 SEMI-FINISHED PRODUCT IN THE MANUFACTURE OF A COMPOSITION FOR SKIN OR HAIR CARE OY GRANULA AB LTD (FI) 2008-02-21 WO disclosed