SCHEMBL16554453

SCHEMBL16554453

CC1(O)CCN(c2nc(N3CCOCC3)nc3c2nnn3Cc2ccccc2Cl)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 18/20 1.00
KDM4E B2RXH2 2/20 0.59
ALDH1A1 P00352 2/20 0.59
GAA P10253 1/20 0.59
MEN1 O00255 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
HTT P42858 1/20 0.56
KMT2A Q03164 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16554610 1.00 CNR2 (1.00) CNR2KDM4EALDH1A1GAAMEN1
SCHEMBL16554450 1.00 CNR2 (1.00) CNR2KDM4EALDH1A1GAAMEN1
SCHEMBL16554727 0.88 CNR2 (1.00) CNR2
SCHEMBL16554731 0.88 CNR2 (1.00) CNR2
SCHEMBL16555005 0.88 CNR2 (1.00) CNR2
SCHEMBL16554959 0.87 CNR2 (1.00) CNR2
SCHEMBL16554976 0.87 CNR2 (1.00) CNR2
SCHEMBL16554965 0.87 CNR2 (1.00) CNR2
SCHEMBL14911410 0.83 CNR2 (0.79) CNR2KDM4EALDH1A1
SCHEMBL14911412 0.83 CNR2 (0.79) CNR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041843-A1 NOVEL TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2016-07-13 EP claimed
WO-2015032769-A1 NOVEL TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2015-03-12 WO claimed
EP-3041843-A1 NOVEL TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2016-07-13 EP disclosed
WO-2015032769-A1 NOVEL TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2015-03-12 WO disclosed