SCHEMBL16587899

SCHEMBL16587899

O=C(NCc1ccccc1)NC[C@H](NC(=O)[C@@H]1CCCCCCCCN1S(=O)(=O)c1ccccc1)C(=O)O

nearest known ligand 0.77

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 10/20 0.77
ITGA2 P17301 7/20 0.77
ITGA4 P13612 1/20 0.77
FKBP1A P62942 5/20 0.60
ITGA5 P08648 3/20 0.54
TDP1 Q9NUW8 1/20 0.53
ITGB3 P05106 1/20 0.53
ITGAV P06756 1/20 0.53
ALDH1A1 P00352 2/20 0.51
MAPK1 P28482 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
TSHR P16473 1/20 0.49
USP2 O75604 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4260019 0.99 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL12084791 0.99 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL8239058 0.96 ITGB1 (0.83) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL12084502 0.96 ITGB1 (0.83) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL4255594 0.96 ITGB1 (0.83) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL1487410 0.93 ITGB1 (0.75) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL12084785 0.92 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL4253400 0.92 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL4253038 0.90 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGA5
SCHEMBL8245501 0.90 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8987306-B2 Inhibitors of integrin alpha2beta1 based on prolyl diaminopropionic acid scaffold THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2015-03-24 US disclosed