SCHEMBL16610380

SCHEMBL16610380

CC(C)CNC(=O)/C=C/c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.51
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NOS3 P29474 2/20 0.45
NOS1 P29475 2/20 0.45
NOS2 P35228 2/20 0.45
HDAC3 O15379 1/20 0.44
ADAM17 P78536 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
HSP90AA1 P07900 1/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28013193 1.00 TRPV1 (0.51) TRPV1HPGDSMN1; SMN2NOS3NOS1
SCHEMBL31345008 0.88 SOAT1 (0.43) TRPV1HPGDSMN1; SMN2NOS3NOS1
SCHEMBL16610377 0.87 MEN1 (0.61) TRPV1HPGDSMN1; SMN2LMNAMEN1
SCHEMBL16610336 0.80 TRPV1 (0.52) TRPV1HPGDSMN1; SMN2PKMKDM4E
SCHEMBL28012614 0.80 TRPV1 (0.52) TRPV1HPGDSMN1; SMN2PKMKDM4E
SCHEMBL16610337 0.79 TRPV1 (0.46) TRPV1HPGDSMN1; SMN2NOS3NOS1
SCHEMBL16610366 0.79 TRPV1 (0.46) TRPV1HPGDSMN1; SMN2NOS3NOS1
SCHEMBL16610365 0.78 TRPV1 (0.50) TRPV1HPGDSMN1; SMN2NOS3NOS1
SCHEMBL28012612 0.78 TRPV1 (0.50) TRPV1HPGDSMN1; SMN2NOS3NOS1
SCHEMBL28663853 0.76 TRPV1 (0.57) TRPV1SMN1; SMN2PKMKDM4EPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed