SCHEMBL16610831

SCHEMBL16610831

Cc1ccc(C(=O)O)c(C)c1.Cc1ccc(C2CCCN2c2nc(C)cc(Nc3ncc(C#N)s3)n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.41
TRPC3 Q13507 1/20 0.34
TRPC6 Q9Y210 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
LCK P06239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610809 0.90 KDR (0.46) KDR
SCHEMBL16610971 0.87 KDR (0.45) KDRTRPC3TRPC6LCK
SCHEMBL16610576 0.82 KDR (0.44) KDRTRPC3TRPC6
SCHEMBL18557099 0.81 KDR (0.43) KDR
SCHEMBL16610520 0.81 KDR (0.40) KDRTRPC3TRPC6
SCHEMBL16610621 0.79 KDR (0.40) KDRTRPC3TRPC6
SCHEMBL18557040 0.79 KDR (0.41) KDR
SCHEMBL16772706 0.78 KDR (0.41) KDRTRPC3TRPC6
SCHEMBL16610755 0.78 KDR (0.41) KDRTRPC3TRPC6
SCHEMBL16610670 0.77 KDR (0.40) KDRTRPC3TRPC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857398-A1 AROMATIC HETEROCYCLIC DERIVATIVE AND PHARMACEUTICAL Nippon Shinyaku Co., Ltd. (JP) 2015-04-08 EP disclosed