SCHEMBL16613104

SCHEMBL16613104

CC1CC[C@@H](C(C)C)[C@H](OC(=O)O[C@@H](C)OC(=O)[C@H]2[C@@H]3C[C@H](F)[C@@](N)(C(=O)O)[C@@H]32)C1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 3/20 0.54
GRM3 Q14832 3/20 0.54
EPHX1 P07099 3/20 0.37
ALDH1A1 P00352 7/20 0.37
HPGD P15428 2/20 0.37
CYP19A1 P11511 2/20 0.34
LMNA P02545 2/20 0.34
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19177419 1.00 GRM2 (0.54) GRM2GRM3EPHX1ALDH1A1HPGD
SCHEMBL16610929 1.00 GRM2 (0.54) GRM2GRM3EPHX1ALDH1A1HPGD
SCHEMBL16610556 1.00 GRM2 (0.54) GRM2GRM3EPHX1ALDH1A1HPGD
SCHEMBL16610461 1.00 GRM2 (0.54) GRM2GRM3EPHX1ALDH1A1HPGD
SCHEMBL16610571 0.96 GRM2 (0.51) GRM2GRM3EPHX1ALDH1A1HPGD
SCHEMBL16610498 0.94 GRM2 (0.51) GRM2GRM3EPHX1ALDH1A1HPGD
SCHEMBL16610463 0.90 GRM2 (0.51) GRM2GRM3ALDH1A1HPGDCYP19A1
SCHEMBL16610610 0.88 GRM2 (0.50) GRM2GRM3ALDH1A1HPGDCYP19A1
SCHEMBL16610573 0.88 GRM2 (0.50) GRM2GRM3EPHX1ALDH1A1HPGD
SCHEMBL19177218 0.87 GRM2 (0.49) GRM2GRM3EPHX1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857385-A1 PRODRUG OF FLUORINE-CONTAINING AMINO ACID Taisho Pharmaceutical Co., Ltd. (JP) 2015-04-08 EP disclosed