SCHEMBL16615259

SCHEMBL16615259

O=C(NCCc1ccccc1)c1cc2c(nn1)NCCN2Cc1cc(F)ccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
POLB P06746 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 5/20 0.41
TP53 P04637 3/20 0.41
TSHR P16473 2/20 0.39
HPGD P15428 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
HIF1A Q16665 1/20 0.38
CCR3 P51677 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615202 0.86 MAPT (0.42) SMN1; SMN2ALDH1A1MAPTTP53
SCHEMBL20859464 0.81 MAPT (0.41) SMN1; SMN2POLBALDH1A1MAPTTP53
SCHEMBL1602177 0.77 MAPT (0.51) GAASMN1; SMN2MAPTTP53NPC1
SCHEMBL17918739 0.70 ALK (0.42) GAAALDH1A1MAPTHPGD
SCHEMBL17918715 0.69 KCNQ2 (0.44) GAAPOLBALDH1A1MAPTTSHR
SCHEMBL16615157 0.69 ALK (0.51) SMN1; SMN2NPC1RAB9ACNR1
SCHEMBL1601988 0.68 ALK (0.50) SMN1; SMN2ALDH1A1MAPTTP53NPC1
SCHEMBL1601557 0.68 ALK (0.75) SMN1; SMN2MAPTTP53
SCHEMBL16615211 0.68 ALK (0.53) ALDH1A1MAPTHPGDNPC1RAB9A
SCHEMBL17918706 0.68 MAPT (0.44) SMN1; SMN2POLBALDH1A1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050884-B1 NEW CHEMICAL COMPOUNDS (DERIVATIVES) AND THEIR APPLICATION FOR THE TREATMENT OF ONCOLOGICAL DISEASES LIMITED LIABILITY COMPANY NATIONAL PHARMACEUTICAL TECH (RU) 2019-04-03 EP disclosed
US-9695182-B2 Chemical compounds (derivatives) and their application for the treatment of oncological diseases LIMITED LIABILITY COMPANY “NATIONAL PHARMACEUTICAL TECHNOLOGIES” (RU) 2017-07-04 US disclosed
US-20160200729-A1 NEW CHEMICAL COMPOUNDS (DERIVATIVES) AND THEIR APPLICATION FOR THE TREATMENT OF ONCOLOGICAL DISEASES LIMITED LIABILITY COMPANY (RU) 2016-07-14 US disclosed
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160200729-A1 NEW CHEMICAL COMPOUNDS (DERIVATIVES) AND THEIR APPLICATION FOR THE TREATMENT OF ONCOLOGICAL DISEASES BRAF, CNKSR1, RAF1 GAA 1401/4885SMN1; SMN2 3750/4885POLB 1072/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.