SCHEMBL16615284

SCHEMBL16615284

CN(C)C1CCN(c2ccc(-c3cc4c(nn3)NCCN4Cc3cc(Cl)ccc3Cl)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 11/20 0.48
JAK2 O60674 2/20 0.40
PRKD3 O94806 2/20 0.40
MAP4K4 O95819 2/20 0.40
ABL1 P00519 2/20 0.40
LCK P06239 2/20 0.40
CSF1R P07333 2/20 0.40
RET P07949 2/20 0.40
MET P08581 2/20 0.40
FGFR1 P11362 2/20 0.40
LTK P29376 2/20 0.40
FLT3 P36888 2/20 0.40
PTK2 Q05397 2/20 0.40
MAP4K2 Q12851 2/20 0.40
NTRK2 Q16620 2/20 0.40
TAOK1 Q7L7X3 2/20 0.40
AURKB Q96GD4 2/20 0.40
MAP4K5 Q9Y4K4 2/20 0.40
CHEK1 O14757 1/20 0.40
AURKA O14965 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17969785 0.88 ALK (0.48) ALKJAK2PRKD3MAP4K4ABL1
SCHEMBL16615294 0.86 ALK (0.44) ALKJAK2PRKD3MAP4K4ABL1
SCHEMBL17918854 0.86 ALK (0.50) ALKJAK2PRKD3MAP4K4ABL1
SCHEMBL17918729 0.84 ALK (0.51) ALKJAK2PRKD3MAP4K4ABL1
SCHEMBL18106058 0.83 ALK (0.41) ALK
SCHEMBL17918707 0.81 ALK (0.41) ALKFGFR1AURKAIGF1RROS1
SCHEMBL17918719 0.77 ALK (0.53) ALKJAK2PRKD3MAP4K4ABL1
SCHEMBL18106065 0.77 ALK (0.39) ALKF10
SCHEMBL17918795 0.76 MAP4K3 (0.35) ALKJAK2METNTRK1MALT1
SCHEMBL17918855 0.75 ALK (0.59) ALKJAK2PRKD3MAP4K4ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9695182-B2 Chemical compounds (derivatives) and their application for the treatment of oncological diseases LIMITED LIABILITY COMPANY “NATIONAL PHARMACEUTICAL TECHNOLOGIES” (RU) 2017-07-04 US disclosed
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed