SCHEMBL1661941

SCHEMBL1661941

COC(=O)CCN1Cc2ccc(-c3nc4ccc(C5(c6ccccc6)C=C5)nc4s3)cc2C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 18/20 0.40
S1PR3 Q99500 7/20 0.37
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
NFKB1 P19838 1/20 0.37
RAB9A P51151 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
S1PR5 Q9H228 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1662151 0.92 NPC1 (0.38) S1PR1S1PR3NPC1PKMHPGD
SCHEMBL1661938 0.90 S1PR1 (0.51) S1PR1S1PR3S1PR5
SCHEMBL1662103 0.84 S1PR1 (0.41) S1PR1S1PR3S1PR5KDM4EALDH1A1
SCHEMBL1662147 0.82 S1PR1 (0.48) S1PR1S1PR3S1PR5
SCHEMBL1662455 0.80 S1PR1 (0.55) S1PR1S1PR3S1PR5
SCHEMBL1664282 0.77 S1PR1 (0.46) S1PR1S1PR3S1PR5
SCHEMBL1662206 0.75 S1PR1 (0.52) S1PR1S1PR3S1PR5
SCHEMBL1662100 0.74 S1PR1 (0.52) S1PR1S1PR3S1PR5
SCHEMBL1661775 0.74 S1PR1 (0.42) S1PR1S1PR3
SCHEMBL1661683 0.72 S1PR1 (0.65) S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2306994-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF Amgen, Inc (US) 2011-04-13 EP disclosed
WO-2009154775-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF AMGEN INC. (US) 2009-12-23 WO disclosed