SCHEMBL16619717

SCHEMBL16619717

COc1cc2c(Nc3cccc(C(O)(C(F)(F)F)C(F)(F)F)c3)c(N)cnc2cc1-c1c(C)noc1C

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 12/20 0.52
CYP2C9 P11712 12/20 0.52
BRD4 O60885 12/20 0.52
BRD2 P25440 9/20 0.52
BRD3 Q15059 9/20 0.52
CYP2C19 P33261 1/20 0.49
PDE4B Q07343 1/20 0.49
EGFR P00533 2/20 0.46
ERBB2 P04626 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16618883 0.86 BRD4 (0.54) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16618707 0.85 CYP3A4 (0.59) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619102 0.82 CYP3A4 (0.48) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619145 0.81 BRD4 (0.54) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619166 0.80 BRD4 (0.53) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16618982 0.79 BRD4 (0.65) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619401 0.78 CYP3A4 (0.58) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619413 0.78 BRD4 (0.77) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16774314 0.78 BRD4 (0.58) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619446 0.77 CYP3A4 (0.78) CYP3A4CYP2C9BRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049629-A1 IMIDAZOQUINOLINE COMPOUNDS AS BROMODOMAIN INHIBITORS Piramal Enterprises Limited (IN) 2015-04-09 WO disclosed