SCHEMBL16619954

SCHEMBL16619954

CNCC(N)c1cnccn1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSP90AA1 P07900 1/20 0.34
PCSK9 Q8NBP7 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
ATM Q13315 1/20 0.31
HPGD P15428 1/20 0.30
AOC1 P19801 1/20 0.30
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1579389 0.79 HSP90AA1 (0.38) KDM4EALDH1A1SMN1; SMN2HSP90AA1ATM
SCHEMBL6278027 0.78 KDM4E (0.46) KDM4EALDH1A1SMN1; SMN2
SCHEMBL6319129 0.78 KDM4E (0.46) KDM4EALDH1A1SMN1; SMN2
SCHEMBL6673370 0.75 KDM4E (0.44) KDM4EALDH1A1SMN1; SMN2PCSK9
SCHEMBL8351769 0.75 HSP90AA1 (0.38) KDM4EALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL16619262 0.75 HSP90AA1 (0.38) KDM4EALDH1A1SMN1; SMN2HSP90AA1ATM
SCHEMBL8230366 0.74 KCNH2 (0.47) ALDH1A1
SCHEMBL4016590 0.71
SCHEMBL2710346 0.71
SCHEMBL266933 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052099-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS Merck Sharp & Dohme Corp. (US) 2016-08-10 EP disclosed
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed