SCHEMBL16620420

SCHEMBL16620420

CC(=O)Nc1cc(C#Cc2cnc3ccc(-c4ccc(C(=O)N5CCN(C(C)(C)C)CC5)cc4)cn23)ccn1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 18/20 0.44
MKNK2 Q9HBH9 18/20 0.44
CYP3A4 P08684 1/20 0.44
EIF4E P06730 4/20 0.43
RIPK2 O43353 1/20 0.40
PIK3C3 Q8NEB9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17969580 0.90 CFTR (0.43) MKNK1MKNK2CYP3A4EIF4ERIPK2
SCHEMBL16620997 0.89 MKNK1 (0.51) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620756 0.83 MKNK1 (0.42) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16621188 0.83 CFTR (0.43) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16621021 0.81 MKNK1 (0.49) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620371 0.81 CFTR (0.43) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620874 0.81 MKNK1 (0.54) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL24520115 0.80 MKNK1 (0.53) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620368 0.79 CFTR (0.42) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620521 0.78 CCNC (0.51) MKNK1MKNK2CYP3A4EIF4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052501-A1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF Agency For Science, Technology And Research (SG) 2016-08-10 EP disclosed
WO-2015050505-A1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-04-09 WO disclosed