SCHEMBL16620514

SCHEMBL16620514

O=C(Nc1ccc(Oc2ccc(B(O)O)cc2)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.56
BRAF P15056 3/20 0.56
MAPK14 Q16539 3/20 0.56
TNNI3K Q59H18 3/20 0.56
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA9 Q16790 1/20 0.53
RAF1 P04049 1/20 0.53
FLT3 P36888 1/20 0.53
TRPV1 Q8NER1 1/20 0.52
CDK8 P49336 2/20 0.51
CDK7 P50613 1/20 0.51
CDK6 Q00534 1/20 0.51
TLR8 Q9NR97 3/20 0.50
EPHX2 P34913 2/20 0.50
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11029731 0.88 TLR8 (0.62) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL11002296 0.84 TLR8 (0.62) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL16628083 0.84 KDR (0.58) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL16621239 0.83 EPHX2 (0.69) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL939205 0.83 KDR (0.79) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL16621127 0.81 MAPT (0.72) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL16621046 0.80 KDR (0.67) KDRBRAFMAPK14TNNI3KCA1
SCHEMBL11012192 0.79 EPHX2 (0.76) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL16628077 0.79 RAF1 (0.67) KDRBRAFMAPK14TNNI3KCA12
SCHEMBL11001590 0.78 EPHX2 (0.81) KDRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051149-A1 SORAFENIB ANALOGS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-04-09 WO disclosed
WO-2015051149-A1 SORAFENIB ANALOGS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-04-09 WO disclosed