SCHEMBL16622905

SCHEMBL16622905

CN1CCN(Cc2cc3c(N4CCOCC4)nc(-c4ccc(NC(=O)Nc5ccc(F)cc5)cc4)nn3c2)CC1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.83
PIK3R1 P27986 3/20 0.74
MTOR P42345 13/20 0.54
PIK3CG P48736 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16727837 0.92 PIK3CA (0.74) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16611561 0.91 PIK3CA (1.00) PIK3CAPIK3R1MTOR
SCHEMBL16727843 0.91 PIK3CA (0.89) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16727838 0.90 PIK3CA (0.84) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16727836 0.88 PIK3CA (0.65) PIK3CAPIK3R1MTOR
SCHEMBL16611050 0.86 PIK3CA (0.72) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL18356848 0.86 PIK3CA (0.81) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16611569 0.85 PIK3CA (1.00) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16727839 0.85 PIK3CA (0.85) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16611681 0.83 PIK3CA (0.86) PIK3CAPIK3R1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857403-A1 PYRROLO[2,1-F][1,2,4]TRIAZINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2015-04-08 EP disclosed