SCHEMBL16622906

SCHEMBL16622906

CCCC1CN(c2nc(-c3ccc(NC(=O)Nc4ccc(F)cc4)cc3)nn3cc(CN4CCN(S(C)(=O)=O)CC4)cc23)CC(C)O1

nearest known ligand 0.73

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 18/20 0.73
PIK3R1 P27986 7/20 0.59
MTOR P42345 6/20 0.46
PIK3CD O00329 1/20 0.43
RAF1 P04049 1/20 0.43
PIK3CB P42338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16611666 0.87 PIK3CA (0.79) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16622901 0.87 PIK3CA (0.79) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16611561 0.84 PIK3CA (1.00) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16622911 0.81 PIK3CA (0.73) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16727836 0.79 PIK3CA (0.65) PIK3CAPIK3R1MTORPIK3CD
SCHEMBL18080823 0.78 PIK3CA (0.65) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16611061 0.78 PIK3CA (0.84) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16611681 0.78 PIK3CA (0.86) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16622899 0.76 PIK3CA (0.81) PIK3CAPIK3R1MTORPIK3CDRAF1
SCHEMBL16611835 0.76 PIK3CA (1.00) PIK3CAPIK3R1MTORPIK3CDRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857403-A1 PYRROLO[2,1-F][1,2,4]TRIAZINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2015-04-08 EP disclosed