SCHEMBL16625807

SCHEMBL16625807

COc1cc(C#Cc2cnc3ccc(-c4ccc(C(=O)N5CCOCC5)c(C)c4)nn23)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 4/20 0.46
MKNK2 Q9HBH9 4/20 0.46
JAK2 O60674 4/20 0.43
JAK1 P23458 4/20 0.43
TYK2 P29597 4/20 0.43
JAK3 P52333 4/20 0.43
EIF4E P06730 2/20 0.43
MTOR P42345 6/20 0.42
PIK3CA P42336 4/20 0.42
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
GSK3A P49840 1/20 0.39
LRRK2 Q5S007 1/20 0.38
ATR Q13535 1/20 0.38
CFTR P13569 1/20 0.37
KIT P10721 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29756374 0.91 MKNK1 (0.56) MKNK1MKNK2EIF4EMTORCFTR
SCHEMBL16620919 0.91 MKNK1 (0.56) MKNK1MKNK2EIF4EMTORCFTR
SCHEMBL17998743 0.89 MTOR (0.48) MKNK1MKNK2JAK2JAK1TYK2
Formic Acid SCHEMBL29756329 0.86 MTOR (0.46) MKNK1MKNK2JAK2JAK1TYK2
Formic Acid SCHEMBL16620929 0.86 MTOR (0.46) MKNK1MKNK2JAK2JAK1TYK2
SCHEMBL16621295 0.81 MKNK1 (0.54) MKNK1MKNK2EIF4E
SCHEMBL16626042 0.81 MKNK1 (0.59) MKNK1MKNK2EIF4EMTORHPGD
SCHEMBL16625832 0.80 MTOR (0.50) MKNK1MKNK2EIF4EMTORPIK3CA
SCHEMBL16620715 0.80 MTOR (0.52) MKNK1MKNK2EIF4EMTORPIK3CA
SCHEMBL29756323 0.79 MKNK1 (0.60) MKNK1MKNK2EIF4EMTORHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050505-A1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-04-09 WO disclosed