SCHEMBL16625990

SCHEMBL16625990

COc1ccc(C#Cc2cnc3ccc(-c4ccc(C(=O)N5CCNCC5)cc4)nn23)cc1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 10/20 0.63
MKNK1 Q9BUB5 9/20 0.63
CYP3A4 P08684 1/20 0.63
EIF4E P06730 3/20 0.53
GRM3 Q14832 4/20 0.47
CCNC P24863 1/20 0.46
CDK8 P49336 1/20 0.46
PARP1 P09874 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
ATR Q13535 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16620923 0.90 MKNK1 (0.63) MKNK2MKNK1CYP3A4EIF4EGRM3
SCHEMBL17998777 0.87 MKNK1 (0.65) MKNK2MKNK1CYP3A4EIF4ECCNC
SCHEMBL20365197 0.83 MKNK1 (0.60) MKNK2MKNK1CYP3A4EIF4ECCNC
SCHEMBL16620734 0.82 MKNK1 (0.60) MKNK2MKNK1CYP3A4EIF4ECCNC
SCHEMBL20365194 0.81 MKNK1 (0.56) MKNK2MKNK1CYP3A4EIF4ECCNC
SCHEMBL17969602 0.80 MKNK1 (0.66) MKNK2MKNK1CYP3A4EIF4E
SCHEMBL16620738 0.79 MKNK1 (0.60) MKNK2MKNK1CYP3A4EIF4E
SCHEMBL29756323 0.79 MKNK1 (0.60) MKNK2MKNK1CYP3A4EIF4E
SCHEMBL16620849 0.79 MKNK1 (0.79) MKNK2MKNK1CYP3A4EIF4E
SCHEMBL16625987 0.79 MKNK1 (0.65) MKNK2MKNK1CYP3A4EIF4EPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050505-A1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-04-09 WO disclosed