SCHEMBL1662661

SCHEMBL1662661

CCc1c(-c2ccccn2)ncc(C)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.47
NPC1 O15118 2/20 0.47
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
LMNA P02545 3/20 0.41
CYP1A2 P05177 2/20 0.41
CCR1 P32246 2/20 0.41
CCR5 P51681 2/20 0.41
CCR8 P51685 2/20 0.41
POLB P06746 1/20 0.41
METAP1 P53582 1/20 0.41
BLM P54132 1/20 0.41
HIF1A Q16665 1/20 0.41
DOHH Q9BU89 1/20 0.41
P4HTM Q9NXG6 1/20 0.41
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CBFB Q13951 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31199032 0.81 KDM4E (0.55) KDM4ENPC1LMNACYP1A2CCR1
SCHEMBL19961977 0.81 KDM4E (0.55) KDM4ENPC1LMNACYP1A2CCR1
SCHEMBL17570275 0.73 KDM4E (0.50) KDM4ENPC1LMNACYP1A2CCR1
SCHEMBL28320230 0.73 KDM4E (0.43) KDM4ENPC1ADORA2AADORA1LMNA
SCHEMBL8962206 0.72 KDM4E (0.42) KDM4ENPC1ADORA2AADORA1LMNA
SCHEMBL3884850 0.72 KDM4E (0.42) KDM4ENPC1ADORA2AADORA1LMNA
SCHEMBL15883898 0.71 SMN1; SMN2 (0.46) KDM4ENPC1LMNACYP1A2CCR1
SCHEMBL30535971 0.70 KDM4E (0.42) KDM4ENPC1LMNACYP1A2CCR1
SCHEMBL4385940 0.70 CYP1A2 (0.42) KDM4ENPC1LMNACYP1A2CCR1
SCHEMBL10957813 0.69 KDM4E (0.58) KDM4ENPC1LMNACYP1A2CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050284-A1 PYRAZOLYLPYRIDINE ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2011-04-28 WO disclosed