SCHEMBL16626820

SCHEMBL16626820

CCOC(=O)c1cnc(NC2(c3ccccc3)CC2)nc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 4/20 0.64
HDAC3 O15379 15/20 0.63
HDAC1 Q13547 15/20 0.63
HDAC2 Q92769 15/20 0.63
HDAC6 Q9UBN7 15/20 0.63
HDAC4 P56524 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC10 Q969S8 1/20 0.57
HDAC11 Q96DB2 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC9 Q9UKV0 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18742534 0.95 HDAC3 (0.65) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL18742411 0.95 HDAC3 (0.65) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL16677936 0.94 HDAC6 (0.67) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL18712282 0.94 HDAC3 (0.65) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL16632207 0.92 HDAC3 (0.55) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL16677935 0.92 HDAC3 (0.55) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL17832599 0.91 HDAC1 (0.62) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL16644384 0.90 HDAC3 (0.66) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL16644382 0.89 HDAC3 (0.70) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL16644404 0.89 HDAC3 (0.69) VNN1HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 67 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025059442-A1 MODULATING PLANT RESPONSES TO STRESS AND GROWTH WITH CHEMICALS REMOTE EPIGENETICS INC. (US) 2025-03-20 WO claimed
EP-4410284-A1 COMPOUND AND METHOD FOR THE TREATMENT OF ZELLWEGER SPECTRUM DISORDER Apteeus (FR) 2024-08-07 EP claimed
US-20230391868-A1 COMPOSITIONS FOR AND METHODS OF TREATING CANCER THE GEORGE WASHINGTON UNIVERSITY 2023-12-07 US claimed
CN-116510024-A Composition, preparation method and application thereof 上海复东生物医药有限责任公司 2023-08-01 CN claimed
CN-114908049-A Use of HDAC6 inhibitors to selectively induce T cell expansion 江苏集萃医学免疫技术研究所有限公司 2022-08-16 CN claimed
US-20260124204-A1 METALLOENZYME INHIBITOR COMPOUNDS EIKONIZO THERAPEUTICS, INC. (US) 2026-05-07 US disclosed
US-12370194-B2 Metalloenzyme inhibitor compounds EIKONIZO THERAPEUTICS, INC. (US) 2025-07-29 US disclosed
WO-2025059442-A1 MODULATING PLANT RESPONSES TO STRESS AND GROWTH WITH CHEMICALS REMOTE EPIGENETICS INC. (US) 2025-03-20 WO disclosed
US-20240307391-A1 METALLOENZYME INHIBITOR COMPOUNDS EIKONIZO THERAPEUTICS, INC. (US) 2024-09-19 US disclosed
CN-115192714-B Use of HDAC6 inhibitors in the manufacture of a medicament for the treatment of DNMT3A gene-deficient cancers 沈阳药科大学 2024-09-17 CN disclosed
WO-2024160990-A1 COMPOUNDS AND METHOD FOR THE TREATMENT OF ZELLWEGER SPECTRUM DISORDER APTEEUS (FR) 2024-08-08 WO disclosed
EP-4410284-A1 COMPOUND AND METHOD FOR THE TREATMENT OF ZELLWEGER SPECTRUM DISORDER Apteeus (FR) 2024-08-07 EP disclosed
US-20150176076-A1 HISTONE DEACETYLASE 6 (HDAC6) BIOMARKERS IN MULTIPLE MYELOMA ACETYLON PHARMACEUTICALS, INC. (US) 2015-06-25 US disclosed
US-20150150871-A1 COMBINATIONS OF HISTONE DEACETYLASE INHIBITORS AND IMMUNOMODULATORY DRUGS ACETYLON PHARMACEUTICALS, INC. (US) 2015-06-04 US disclosed
US-20150105358-A1 COMBINATIONS OF HISTONE DEACETYLASE INHIBITORS AND IMMUNOMODULATORY DRUGS ACETYLON PHARMACEUTICALS, INC. (US) 2015-04-16 US disclosed
US-20150105383-A1 HDAC Inhibitors, Alone Or In Combination With PI3K Inhibitors, For Treating Non-Hodgkin's Lymphoma ACETYLON PHARMACEUTICALS, INC. (US) 2015-04-16 US disclosed
WO-2015054197-A1 HDAC INHIBITORS, ALONE OR IN COMBINATION WITH BTK INHIBITORS, FOR TREATING NON-HODGKIN'S LYMPHOMA ACETYLON PHARMACEUTICALS, INC. (US) 2015-04-16 WO disclosed
US-20150105409-A1 HDAC INHIBITORS, ALONE OR IN COMBINATION WITH BTK INHIBITORS, FOR TREATING NONHODGKIN'S LYMPHOMA Acetylon Pharmaceticals, Inc. (US) 2015-04-16 US disclosed
WO-2015054175-A1 COMBINATIONS OF HISTONE DEACTYLASE INHIBITORS AND IMMUNOMODULATORY DRUGS ACETYLON PHARMACEUTICALS, INC. (US) 2015-04-16 WO disclosed
US-20150099744-A1 COMBINATIONS OF HISTONE DEACETYLASE INHIBITORS AND EITHER HER2 INHIBITORS OR PI3K INHIBITORS ACETYLON PHARMACEUTICALS, INC. (US) 2015-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150105409-A1 HDAC INHIBITORS, ALONE OR IN COMBINATION WITH BTK INHIBITORS, FOR TREATING NONHODGKIN'S LYMPHOMA BTK, HDAC2, HDAC5 VNN1 1989/4885HDAC3 10/4885HDAC1 8/4885
US-20240307391-A1 METALLOENZYME INHIBITOR COMPOUNDS HDAC6, HDAC1, HDAC2 VNN1 1112/4885HDAC3 7/4885HDAC1 2/4885
US-20150150871-A1 COMBINATIONS OF HISTONE DEACETYLASE INHIBITORS AND IMMUNOMODULATORY DRUGS HDAC5, HDAC4, HDAC3 VNN1 1405/4885HDAC3 3/4885HDAC1 5/4885
US-20230391868-A1 COMPOSITIONS FOR AND METHODS OF TREATING CANCER CD47, HDAC6, HDAC3 VNN1 3761/4885HDAC3 3/4885HDAC1 4/4885
US-20150105383-A1 HDAC Inhibitors, Alone Or In Combination With PI3K Inhibitors, For Treating Non-Hodgkin's Lymphoma HDAC5, HDAC9, HDAC4 VNN1 1346/4885HDAC3 8/4885HDAC1 5/4885
US-20150099744-A1 COMBINATIONS OF HISTONE DEACETYLASE INHIBITORS AND EITHER HER2 INHIBITORS OR PI3K INHIBITORS HDAC6, HDAC2, HDAC5 VNN1 1446/4885HDAC3 7/4885HDAC1 6/4885
US-20260124204-A1 METALLOENZYME INHIBITOR COMPOUNDS HDAC6, HDAC3, HDAC1 VNN1 2427/4885HDAC3 2/4885HDAC1 3/4885
US-20150176076-A1 HISTONE DEACETYLASE 6 (HDAC6) BIOMARKERS IN MULTIPLE MYELOMA HDAC5, HDAC6, HDAC9 VNN1 2171/4885HDAC3 8/4885HDAC1 7/4885
US-20150105358-A1 COMBINATIONS OF HISTONE DEACETYLASE INHIBITORS AND IMMUNOMODULATORY DRUGS HDAC5, HDAC4, HDAC2 VNN1 1312/4885HDAC3 6/4885HDAC1 5/4885
US-12370194-B2 Metalloenzyme inhibitor compounds HDAC6, HDAC1, HDAC2 VNN1 1112/4885HDAC3 7/4885HDAC1 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.