SCHEMBL16629060

SCHEMBL16629060

COc1cnc(-n2cnc(C)n2)c2[nH]cc(C(=O)C(=O)NCC3CN(C(=O)OC(C)(C)C)C3)c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C8 P10632 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2B6 P20813 1/20 0.53
CYP2C19 P33261 1/20 0.53
KCNH2 Q12809 1/20 0.53
NAMPT P43490 1/20 0.37
JAK3 P52333 1/20 0.34
BTK Q06187 2/20 0.33
LMNA P02545 3/20 0.32
TP53 P04637 3/20 0.32
GPR119 Q8TDV5 3/20 0.32
EGLN2 Q96KS0 1/20 0.32
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16629074 0.89 CYP3A4 (0.54) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL16618926 0.86 CYP2C9 (0.71) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL9914945 0.83 CYP3A4 (0.72) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL2629197 0.77 CYP3A4 (0.65) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL14754253 0.76 CYP3A4 (0.67) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL1473305 0.76 CYP3A4 (0.68) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
Hydrochloric Acid SCHEMBL1472468 0.75 CYP3A4 (0.67) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL17954534 0.74 CYP3A4 (0.62) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL14754234 0.73 CYP3A4 (0.65) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6
SCHEMBL9914944 0.73 CYP3A4 (0.75) CYP3A4CYP2C9CYP1A2CYP2C8CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9920073-B2 Compositions useful for inhibiting HIV-1 infection and methods using same DREXEL UNIVERSITY (US) 2018-03-20 US disclosed
WO-2015051230-A1 NOVEL COMPOSITIONS USEFUL FOR INHIBITING HIV-1 INFECTION AND METHODS USING SAME DREXEL UNIVERSITY (US) 2015-04-09 WO disclosed