SCHEMBL16629061

SCHEMBL16629061

CS(=O)(=O)NCCCNCl

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
POLB P06746 1/20 0.44
MAPT P10636 2/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA12 O43570 1/20 0.37
CA7 P43166 1/20 0.37
CA14 Q9ULX7 1/20 0.37
GRIA1 P42261 3/20 0.34
RECQL P46063 2/20 0.33
ALOX15 P16050 1/20 0.32
PPARA Q07869 2/20 0.32
NQO2 P16083 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12090531 0.81 POLB (0.52) ALDH1A1POLBMAPTCA1CA2
SCHEMBL14740296 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL14739816 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL15836237 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL14739086 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL14739515 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL14739265 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL14740061 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL14740248 0.78 GRIA1 (0.52) ALDH1A1POLBCA1CA2CA12
SCHEMBL2582338 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9751888-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-09-05 US disclosed
US-20160222016-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2016-08-04 US disclosed
WO-2015051241-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160222016-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB ALDH1A1 3154/4885POLB 1743/4885MAPT 1605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.