SCHEMBL16630638

SCHEMBL16630638

COc1ccc(CN(C)C(=O)c2ccc(C[C@@H]3CC[C@H](Cc4ccc(Cl)nc4)N3)cc2)cn1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 2/20 0.39
PSEN2 P49810 2/20 0.39
APH1B Q8WW43 2/20 0.39
NCSTN Q92542 2/20 0.39
APH1A Q96BI3 2/20 0.39
PSENEN Q9NZ42 2/20 0.39
TAS2R14 Q9NYV8 1/20 0.38
CCNE1 P24864 3/20 0.36
CDK2 P24941 3/20 0.36
GSK3B P49841 2/20 0.36
OXTR P30559 1/20 0.36
AGTR2 P50052 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
JAK2 O60674 1/20 0.34
PDK1 Q15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16619861 0.88 ADRB3 (0.38)
SCHEMBL16619863 0.88 ADRB3 (0.38)
SCHEMBL16619204 0.81 ADRB3 (0.49)
SCHEMBL16619207 0.81 ADRB3 (0.49)
SCHEMBL16619973 0.80 ADRB3 (0.42)
SCHEMBL16619975 0.80 ADRB3 (0.42)
SCHEMBL16619277 0.78 ADRB3 (0.50)
SCHEMBL16619276 0.78 ADRB3 (0.50)
SCHEMBL16619775 0.77 ADRB3 (0.43)
SCHEMBL16619777 0.77 ADRB3 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed