SCHEMBL16630758

SCHEMBL16630758

CC(=N)n1cc(CN(C)C(=O)c2ccc(C[C@@H]3CC[C@H]([C@H](O)c4ccc(Cl)nc4)N3)cc2)ccc1=N

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 19/20 0.37
SLC6A2 P23975 3/20 0.37
KCNH2 Q12809 8/20 0.36
ADRB2 P07550 5/20 0.36
SLC6A4 P31645 3/20 0.35
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16630773 0.87 ADRB3 (0.49) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619973 0.87 ADRB3 (0.42) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619975 0.87 ADRB3 (0.42) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619851 0.84 ADRB3 (0.38) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619853 0.84 ADRB3 (0.38) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL18019667 0.84 ADRB3 (0.40) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619861 0.82 ADRB3 (0.38) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619863 0.82 ADRB3 (0.38) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619620 0.82 ADRB3 (0.40) ADRB3SLC6A2KCNH2ADRB2SLC6A4
SCHEMBL16619622 0.82 ADRB3 (0.40) ADRB3SLC6A2KCNH2ADRB2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed