SCHEMBL16638818

SCHEMBL16638818

C[C@@H](O)[C@@H](CO[Si](C)(C)C(C)(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA7 P43166 2/20 0.49
CYP2D6 P10635 1/20 0.41
CTSK P43235 8/20 0.38
KMT2A Q03164 1/20 0.37
CTSS P25774 3/20 0.37
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA4 P22748 1/20 0.36
CA9 Q16790 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GLS O94925 1/20 0.34
KLK5 Q9Y337 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2497438 1.00 CA1 (0.49) CA1CA2CA7CYP2D6CTSK
SCHEMBL15215101 1.00 CA1 (0.49) CA1CA2CA7CYP2D6CTSK
SCHEMBL16317020 0.90 CA1 (0.58) CA1CA2CA7CYP2D6CTSK
SCHEMBL2492647 0.87 CA1 (0.48) CA1CA2CA7CYP2D6CTSK
SCHEMBL12191651 0.87 CA1 (0.48) CA1CA2CA7CYP2D6CTSK
SCHEMBL26748578 0.85 CA1 (0.45) CA1CA2CA7CYP2D6CTSK
SCHEMBL3198135 0.85 CA1 (0.42) CA1CA2CA7CYP2D6CTSK
SCHEMBL16690443 0.83 CYP2D6 (0.47) CA1CA2CA7CYP2D6CTSK
SCHEMBL16690460 0.83 CA1 (0.44) CA1CA2CA7CYP2D6CTSK
SCHEMBL5001764 0.83 CA1 (0.45) CA1CA2CA7CYP2D6CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2540720-B1 1,3,4,8-TETRAHYDRO-2H-PYRIDO[1,2-A]PYRAZINE DERIVATIVE AND USE OF SAME AS HIV INTEGRASE INHIBITOR JAPAN TOBACCO INC (JP) 2015-04-15 EP disclosed