SCHEMBL16639149

SCHEMBL16639149

Cc1nc2ccccc2nc1-c1cc2nc(N3CC[C@H](F)C3)cc(N)n2n1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 13/20 0.70
PDE6D O43924 1/20 0.56
PDE5A O76074 1/20 0.56
PDE6A P16499 1/20 0.56
PDE6G P18545 1/20 0.56
PDE4A P27815 1/20 0.56
PDE6B P35913 1/20 0.56
PDE6C P51160 1/20 0.56
PDE4B Q07343 1/20 0.56
PDE4C Q08493 1/20 0.56
PDE4D Q08499 1/20 0.56
PDE6H Q13956 1/20 0.56
ALDH1A1 P00352 3/20 0.40
NPC1 O15118 2/20 0.40
HPGD P15428 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NFKB1 P19838 1/20 0.40
HTT P42858 1/20 0.40
NFKB2 Q00653 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6900533 0.88 PDE10A (0.71) PDE10APDE6DPDE5APDE6APDE6G
SCHEMBL14211805 0.85 PDE10A (0.73) PDE10APDE6DPDE5APDE6APDE6G
SCHEMBL6899512 0.85 PDE10A (0.54) PDE10AALDH1A1NPC1HPGDRAB9A
SCHEMBL14120049 0.84 PDE10A (0.66) PDE10APDE6DPDE5APDE6APDE6G
SCHEMBL6899491 0.84 PDE10A (0.69) PDE10APDE6DPDE5APDE6APDE6G
SCHEMBL14211793 0.84 PDE10A (0.69) PDE10APDE6DPDE5APDE6APDE6G
SCHEMBL14211803 0.84 PDE10A (0.72) PDE10APDE6DPDE5APDE6APDE6G
SCHEMBL14119732 0.84 PDE10A (0.72) PDE10APDE6DPDE5APDE6APDE6G
SCHEMBL6900869 0.83 PDE10A (1.00) PDE10APDE6DPDE5APDE6APDE6G
Hydrochloric Acid SCHEMBL14119954 0.83 PDE10A (0.73) PDE10APDE6DPDE5APDE6APDE6G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2539342-B1 PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS PDE10 INHIBITORS MITSUBISHI TANABE PHARMA CORP (JP) 2015-04-15 EP disclosed